Logo: to the web site of Uppsala University

uu.sePublications from Uppsala University
Change search
CiteExportLink to record
Permanent link

Direct link
Cite
Citation style
  • apa
  • ieee
  • modern-language-association
  • vancouver
  • Other style
More styles
Language
  • de-DE
  • en-GB
  • en-US
  • fi-FI
  • nn-NO
  • nn-NB
  • sv-SE
  • Other locale
More languages
Output format
  • html
  • text
  • asciidoc
  • rtf
Role of FKBP5 in adipose tissue function: Implications for obesity and insulin sensitivity
Uppsala University, Disciplinary Domain of Medicine and Pharmacy, Faculty of Medicine, Department of Medical Sciences, Clinical diabetology and metabolism.ORCID iD: 0000-0003-2016-665X
Uppsala University, Disciplinary Domain of Medicine and Pharmacy, Faculty of Medicine, Department of Medical Sciences, Clinical diabetology and metabolism.ORCID iD: 0000-0002-0964-6700
Uppsala University, Disciplinary Domain of Medicine and Pharmacy, Faculty of Medicine, Department of Medical Sciences, Clinical diabetology and metabolism.ORCID iD: 0000-0003-0200-0760
Uppsala University, Disciplinary Domain of Medicine and Pharmacy, Faculty of Medicine, Department of Medical Sciences, Clinical diabetology and metabolism.ORCID iD: 0000-0001-9348-4603
Show others and affiliations
2026 (English)In: Molecular and Cellular Endocrinology, ISSN 0303-7207, E-ISSN 1872-8057, Vol. 613, article id 112718Article in journal (Refereed) Published
Abstract [en]

FK506-binding protein 51 (FKBP51, encoded by the FKBP5 gene) is a key regulator of glucocorticoid signaling and has been implicated in metabolism and insulin sensitivity, but its specific role in human adipose tissue remains unclear. This study investigated the role of FKBP51 in human adipose tissue and its impact on glucose metabolism and insulin signaling. FKBP5 was measured in paired subcutaneous (SAT) and omental (OAT) adipose tissue samples from 56 subjects with and without obesity, and in SAT from individuals with obesity during weight loss up to 104 weeks post-bariatric surgery. Furthermore, FKBP51 knockdown adipocytes were used to study its effects on insulin signaling and glucose uptake. FKBP5 gene expression, but not protein expression, was significantly lower in obese individuals in both SAT and OAT compared to lean and overweight subjects, and it inversely correlated with insulin resistance measured by homeostatic model assessment of insulin resistance (HOMA-IR). After bariatric surgery, FKBP5 expression in SAT increased to levels similar to those in non-obese controls. Knockdown of FKBP5 in human adipocytes reduced GLUT1 gene expression and insulin-stimulated AKT Ser473 phosphorylation, however, maximal insulin-stimulated glucose uptake rate remained unchanged. Our findings suggest that FKBP5 levels in adipose tissue are reduced in obesity, and this decrease impairs insulin signaling in adipocytes without altering maximal glucose capacity, indicating a limited effect on glucose uptake under the tested conditions.

Place, publisher, year, edition, pages
Elsevier, 2026. Vol. 613, article id 112718
Keywords [en]
Obesity, Weight loss, FKBP5, Adiposity, Glucocorticoids, Metabolism
National Category
Endocrinology and Diabetes Cell and Molecular Biology
Identifiers
URN: urn:nbn:se:uu:diva-576213DOI: 10.1016/j.mce.2025.112718ISI: 001650131000001PubMedID: 41397645Scopus ID: 2-s2.0-105025408668OAI: oai:DiVA.org:uu-576213DiVA, id: diva2:2029141
Funder
Swedish Research Council, 2024-03344Swedish Foundation for Strategic Research, CMP22-0014Available from: 2026-01-16 Created: 2026-01-16 Last updated: 2026-01-16Bibliographically approved

Open Access in DiVA

fulltext(5920 kB)182 downloads
File information
File name FULLTEXT01.pdfFile size 5920 kBChecksum SHA-512
7752412eb59659ffefb99c4f05793ead3627831f89a6038e72659dc1a7cfffb00566c563e81c003176a0e74beeb933cc64fad70a50e6690125f49c8e0fb3d1d2
Type fulltextMimetype application/pdf

Other links

Publisher's full textPubMedScopus

Authority records

Laterveer, RutgerHetty, SusanneMathioudaki, ArgyriLundqvist, Martin H.Svensson, Maria K.Sundbom, MagnusKatsogiannos, PetrosEriksson, JanPereira, Maria J.

Search in DiVA

By author/editor
Laterveer, RutgerHetty, SusanneMathioudaki, ArgyriLundqvist, Martin H.Svensson, Maria K.Sundbom, MagnusKatsogiannos, PetrosEriksson, JanPereira, Maria J.
By organisation
Clinical diabetology and metabolismRenal MedicineUppsala Clinical Research Center (UCR)Upper Abdominal Surgery
In the same journal
Molecular and Cellular Endocrinology
Endocrinology and DiabetesCell and Molecular Biology

Search outside of DiVA

GoogleGoogle Scholar
The number of downloads is the sum of all downloads of full texts. It may include eg previous versions that are now no longer available

doi
pubmed
urn-nbn

Altmetric score

doi
pubmed
urn-nbn
Total: 1000 hits
CiteExportLink to record
Permanent link

Direct link
Cite
Citation style
  • apa
  • ieee
  • modern-language-association
  • vancouver
  • Other style
More styles
Language
  • de-DE
  • en-GB
  • en-US
  • fi-FI
  • nn-NO
  • nn-NB
  • sv-SE
  • Other locale
More languages
Output format
  • html
  • text
  • asciidoc
  • rtf